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Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50017206
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179048((2S,3S,4R,5R)-3,4-Dihydroxy-5-{6-[3-(4-sulfamoyl-p...)
Affinity DataKi:  9.73nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179051(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  16.3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179022(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  17.1nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179027(1-(4-acetylphenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  20.9nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179023(1-benzyl-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  38.3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179030((2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(pyridin-2-...)
Affinity DataKi:  54.1nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179041(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  77.6nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179049(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  89.5nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179047(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179037(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  149nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179031(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  154nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179029((2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(5-methyl-i...)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179038((2S,3S,4R,5R)-5-(6-(2-(2,4-dichlorophenyl)acetamid...)
Affinity DataKi:  167nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179052((2S,3S,4R,5R)-5-(6-{bis[(4-nitrophenyl)carbamoyl]a...)
Affinity DataKi:  168nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179034(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  211nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179043(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179050(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  315nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179026(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  319nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179036(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  324nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179044((2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-{3-[4-(pyrimidin-...)
Affinity DataKi:  405nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179046(1-(3,4-dimethoxyphenethyl)-3-(9-((2R,3R,4S,5S)-5-(...)
Affinity DataKi:  411nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179039(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  532nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179028(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  581nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179045(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  611nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179032(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  696nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179042(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  713nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179033((2S,3S,4R,5R)-5-(6-(2-chlorobenzamido)-9H-purin-9-...)
Affinity DataKi:  754nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179053((2S,3S,4R,5R)-5-(6-benzamido-9H-purin-9-yl)-N-ethy...)
Affinity DataKi:  824nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179024((2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-methox...)
Affinity DataKi:  837nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179025((2S,3S,4R,5R)-5-{6-[(Biphenyl-4-carbonyl)-amino]-p...)
Affinity DataKi:  979nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179040(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  5.55E+3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
Vigo University

Curated by ChEMBL
LigandPNGBDBM50179035((2S,3S,4R,5R)-5-(6-{bis[(5-chloropyridin-2-yl)carb...)
Affinity DataKi:  5.70E+3nMAssay Description:Displacement of [125I]AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed