Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50019026
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200937(estradiol 3-O-sulfamate | CHEMBL219321)
Affinity DataIC50: 16nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50159804(estradiol 3,17-O,O-bis-sulfamate | sulfamic acid (...)
Affinity DataIC50: 18nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200936(2-Methoxyestradiol-3,17-O,O-bis-sulfamate | 2-meth...)
Affinity DataIC50: 39nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50134329(Sulfamic acid (8R,9S,13S,14S)-13-methyl-17-oxo-7,8...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human CA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200942(3-O-sulfamoylestradiol 17beta-O-(N,N-dipentyl)sulf...)
Affinity DataIC50: 190nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200939(2-methylsulfanylestradiol 3,17-O,O-bis-sulfamate |...)
Affinity DataIC50: 320nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200936(2-Methoxyestradiol-3,17-O,O-bis-sulfamate | 2-meth...)
Affinity DataIC50: 379nMAssay Description:Inhibition of human CA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200940(2-methoxyestradiol 17-O-sulfamate | (13ALPHA,14BET...)
Affinity DataIC50: 526nMAssay Description:Inhibition of human CA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200941((9BETA,13ALPHA,14BETA,17ALPHA)-2-ETHYLESTRA-1(10),...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50200938(estradiol 17-O-sulfamate | CHEMBL220493)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of STS in placental microsomes by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed