Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50030683
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300112(trans-1-cyclopentyl-6-(4-methyl-1-(quinoxalin-6-yl...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300112(trans-1-cyclopentyl-6-(4-methyl-1-(quinoxalin-6-yl...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300099(6-benzyl-1-cyclopentyl-1,5-dihydro-4H-pyrazolo[3,4...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300099(6-benzyl-1-cyclopentyl-1,5-dihydro-4H-pyrazolo[3,4...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300099(6-benzyl-1-cyclopentyl-1,5-dihydro-4H-pyrazolo[3,4...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50300099(6-benzyl-1-cyclopentyl-1,5-dihydro-4H-pyrazolo[3,4...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50300107(trans-1-cyclopentyl-6-(4-methyl-1-((2-methylpyrimi...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300109(trans-1-cyclopentyl-6-(1-((1,3-dimethyl-1H-pyrazol...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300110(trans-1-cyclopentyl-6-(4-methyl-1-((5-methylisoxaz...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300111(trans-1-cyclopentyl-6-(1-(imidazo[1,2-a]pyridin-2-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300111(trans-1-cyclopentyl-6-(1-(imidazo[1,2-a]pyridin-2-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300108(trans-1-cyclopentyl-6-(4-methyl-1-((5-methylpyrazi...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300106(trans-1-cyclopentyl-6-(4-methyl-1-((6-(trifluorome...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300105(trans-1-cyclopentyl-6-(1-((6-methoxypyridin-3-yl)m...)
Affinity DataIC50: 29nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300103(trans-1-cyclopentyl-6-(4-methyl-1-(3-methylbenzyl)...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300103(trans-1-cyclopentyl-6-(4-methyl-1-(3-methylbenzyl)...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300102(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-cyclo...)
Affinity DataIC50: 63nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300102(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-cyclo...)
Affinity DataIC50: 63nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300101(6-[(3S,4S)-1-benzyl-4-methylpyrrolidin-3-yl]-1-(1-...)
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50300101(6-[(3S,4S)-1-benzyl-4-methylpyrrolidin-3-yl]-1-(1-...)
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50300112(trans-1-cyclopentyl-6-(4-methyl-1-(quinoxalin-6-yl...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300112(trans-1-cyclopentyl-6-(4-methyl-1-(quinoxalin-6-yl...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300110(trans-1-cyclopentyl-6-(4-methyl-1-((5-methylisoxaz...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300100(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-isobu...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300100(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-isobu...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300106(trans-1-cyclopentyl-6-(4-methyl-1-((6-(trifluorome...)
Affinity DataIC50: 195nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300109(trans-1-cyclopentyl-6-(1-((1,3-dimethyl-1H-pyrazol...)
Affinity DataIC50: 195nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300104(trans-1-cyclopentyl-6-(4-methyl-1-(pyridin-2-ylmet...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300104(trans-1-cyclopentyl-6-(4-methyl-1-(pyridin-2-ylmet...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant PDE9A expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300108(trans-1-cyclopentyl-6-(4-methyl-1-((5-methylpyrazi...)
Affinity DataIC50: 209nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300111(trans-1-cyclopentyl-6-(1-(imidazo[1,2-a]pyridin-2-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300111(trans-1-cyclopentyl-6-(1-(imidazo[1,2-a]pyridin-2-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300105(trans-1-cyclopentyl-6-(1-((6-methoxypyridin-3-yl)m...)
Affinity DataIC50: 269nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 349nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300107(trans-1-cyclopentyl-6-(4-methyl-1-((2-methylpyrimi...)
Affinity DataIC50: 407nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300103(trans-1-cyclopentyl-6-(4-methyl-1-(3-methylbenzyl)...)
Affinity DataIC50: 563nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300103(trans-1-cyclopentyl-6-(4-methyl-1-(3-methylbenzyl)...)
Affinity DataIC50: 563nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300102(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-cyclo...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300102(trans-6-(1-benzyl-4-methylpyrrolidin-3-yl)-1-cyclo...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE3AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE4CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE7BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300113(1-cyclopentyl-6-[(3S,4S)-4-methyl-1-(quinoxalin-6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PDE11More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50300104(trans-1-cyclopentyl-6-(4-methyl-1-(pyridin-2-ylmet...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant PDE1C expressed in Sf9 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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