Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50031076
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50206624(3-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-4-hyd...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306574(2-(4-Adamantan-1-yl-phenoxy)-N-[2-hydroxy-5-(4,4,5...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306575((3-{2-[4-(adamantan-1-yl)phenoxy]acetamido}-4-hydr...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306568(2-(4-tert-butylphenoxy)-N-(2-hydroxy-5-(4,4,5,5-te...)
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306573(3-(2-(4-tert-butylphenoxy)acetamido)-4-hydroxyphen...)
Affinity DataIC50: 4.03E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306567(2-(4-cyclohexylphenoxy)-N-(2-hydroxy-5-(4,4,5,5-te...)
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306572(3-(2-(4-cyclohexylphenoxy)acetamido)-4-hydroxyphen...)
Affinity DataIC50: 8.48E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306564(N-(2-hydroxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxabor...)
Affinity DataIC50: 9.06E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306565(2-(4-ethylphenoxy)-N-(2-hydroxy-5-(4,4,5,5-tetrame...)
Affinity DataIC50: 9.18E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306566(2-(biphenyl-4-yloxy)-N-(2-hydroxy-5-(4,4,5,5-tetra...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306569(4-hydroxy-3-(2-(p-tolyloxy)acetamido)phenylboronic...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306570(3-(2-(4-ethylphenoxy)acetamido)-4-hydroxyphenylbor...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Gakushuin University

Curated by ChEMBL
LigandPNGBDBM50306571(3-(2-(biphenyl-4-yloxy)acetamido)-4-hydroxyphenylb...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hypoxia-induced HIF1alpha activation in human HeLa cells after 12 hrs by HRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed