Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50034009
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50134329(Sulfamic acid (8R,9S,13S,14S)-13-methyl-17-oxo-7,8...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human purified steroid sulfataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM13058(6-oxo-6,7,8,9,10,11-hexahydrocyclohepta[c]chromen-...)
Affinity DataIC50: 350nMAssay Description:Inhibition of steroid sulfatase in human intact MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human purified steroid sulfataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355361(CHEMBL1835541)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355369(CHEMBL1627935)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355367(CHEMBL1835539)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355366(CHEMBL1835538)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355368(CHEMBL1835540)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355370(CHEMBL1835542)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355371(CHEMBL1835543)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50311659((8R,9S,13S,14S)-2-bromo-3-hydroxy-13-methyl-7,8,9,...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM17289(folliculin | (1S,10R,11S,15S)-5-hydroxy-15-methylt...)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355364(CHEMBL1835632)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355365(CHEMBL1835537)
Affinity DataIC50: 2.15E+5nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355373(CHEMBL1835545)
Affinity DataIC50: 2.24E+5nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  30nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  85nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355362(CHEMBL1835544)
Affinity DataKi:  90nMAssay Description:Mixed type inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355372(CHEMBL482212)
Affinity DataKi:  250nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355361(CHEMBL1835541)
Affinity DataKi:  1.40E+3nMAssay Description:Non-Competitive inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Reversible inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355363(CHEMBL1835424)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate after 5 mins by Kitz-Wilson plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetSteryl-sulfatase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50355360(CHEMBL1835425)
Affinity DataKi:  8.50E+4nMAssay Description:Reversible inhibition of human steroid sulfatase using 4-methylumbelliferyl sulfate substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed