Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50035138
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(GDP-Azasugar analogue | CHEMBL52741)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 1 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM92459(Guanosine Diphosphate | CHEMBL384759 | GDP)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(GDP-Azasugar analogue | CHEMBL52741)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101907(({[(2R,3S,4R,5R)-5-(2-azaniumyl-6-hydroxy-9H-purin...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101906(GDP-Azasugar analogue | CHEMBL53188)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed