Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50036054
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001273(CHEMBL124095 | 3-((2-Carbamoyl-ethylsulfanyl)-{3-[...)
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001285(3-(((3-(2-(7-chloroquinoline-2-yl)ethenyl)phenyl)(...)
Affinity DataIC50: 0.800nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001293(CHEMBL408753 | 3-[{3-[2-(7-Chloro-quinolin-2-yl)-v...)
Affinity DataIC50: 2.20nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230047(CHEMBL127877)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001296(CHEMBL125135 | 3-{(2-Carboxy-ethylsulfanyl)-[3-(7-...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230045(CHEMBL340726)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001271(CHEMBL444331 | 3-((2-Carboxy-ethylsulfanyl)-{3-[2-...)
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230044(CHEMBL123577)
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230074(CHEMBL126859)
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001269(CHEMBL123623 | 3-((2-Carboxy-ethylsulfanyl)-{3-[2-...)
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001288(CHEMBL124259 | 3-[{3-[2-(7-Chloro-quinolin-2-yl)-v...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001289(CHEMBL123958 | 3-{(2-Dimethylcarbamoyl-ethylsulfan...)
Affinity DataIC50: 89nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230078(CHEMBL128010)
Affinity DataIC50: 97nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001300(CHEMBL339713 | 3-((2-Carboxy-ethylsulfanyl)-{3-[3-...)
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230046(CHEMBL125799)
Affinity DataIC50: 270nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001295(CHEMBL338166 | dilithium; 3-((2-carboxy-ethylsulfa...)
Affinity DataIC50: 440nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230049(CHEMBL125027)
Affinity DataIC50: 480nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230043(CHEMBL125978)
Affinity DataIC50: 495nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50012434(1-[3-(Quinolin-2-ylmethoxy)-phenyl]-hexan-1-ol | 1...)
Affinity DataIC50: 510nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230077(CHEMBL414242)
Affinity DataIC50: 560nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230042(CHEMBL127530)
Affinity DataIC50: 580nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001282(CHEMBL124741 | {3-[2-(6-Methyl-quinolin-2-yl)-viny...)
Affinity DataIC50: 930nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230075(CHEMBL126379)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230051(CHEMBL125139)
Affinity DataIC50: 1.43E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230052(CHEMBL124760)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230050(CHEMBL124709)
Affinity DataIC50: 1.78E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001280(CHEMBL338876 | 2-(2-Pyridin-4-yl-vinyl)-quinoline)
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001290(trans-2-styrylquinoline | CHEMBL127579 | cid_53574...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001283(CHEMBL127816 | 2-(2-Pyridin-3-yl-vinyl)-quinoline)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230048(CHEMBL127905)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50001270(CHEMBL127545 | 2-(2-(quinolin-2-yl)vinyl)phenol | ...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50230076(CHEMBL339304)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed