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Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50036644
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50369386(CHEMBL608327)
Affinity DataKi:  0.330nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179025((2S,3S,4R,5R)-5-{6-[(Biphenyl-4-carbonyl)-amino]-p...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179048((2S,3S,4R,5R)-3,4-Dihydroxy-5-{6-[3-(4-sulfamoyl-p...)
Affinity DataKi:  9.70nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  10nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179051(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  16nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179038((2S,3S,4R,5R)-5-(6-(2-(2,4-dichlorophenyl)acetamid...)
Affinity DataKi:  16nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179022(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  17nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50455117(CHEMBL2113550)
Affinity DataKi:  17nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179027(1-(4-acetylphenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  21nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179022(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  22nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179038((2S,3S,4R,5R)-5-(6-(2-(2,4-dichlorophenyl)acetamid...)
Affinity DataKi:  27nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179043(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  29nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179023(1-benzyl-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  38nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  54nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50455116(CHEMBL2113540)
Affinity DataKi:  54nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  56nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179022(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  59nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179027(1-(4-acetylphenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  73nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179036(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  75nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179041(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  78nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179024((2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-methox...)
Affinity DataKi:  86nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179052((2S,3S,4R,5R)-5-(6-{bis[(4-nitrophenyl)carbamoyl]a...)
Affinity DataKi:  89nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179041(1-(2-chloro-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  90nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179049(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  90nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179050(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  103nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179047(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  107nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  113nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179037(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  129nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179039(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  146nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179037(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  149nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179031(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  154nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50369388(CHEMBL610112)
Affinity DataKi:  155nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179038((2S,3S,4R,5R)-5-(6-(2-(2,4-dichlorophenyl)acetamid...)
Affinity DataKi:  167nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179052((2S,3S,4R,5R)-5-(6-{bis[(4-nitrophenyl)carbamoyl]a...)
Affinity DataKi:  168nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179023(1-benzyl-3-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,...)
Affinity DataKi:  171nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179040(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  208nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179034(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  211nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179024((2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-methox...)
Affinity DataKi:  237nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179047(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  247nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179043(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  251nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179053((2S,3S,4R,5R)-5-(6-benzamido-9H-purin-9-yl)-N-ethy...)
Affinity DataKi:  252nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179047(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  255nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179043(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  260nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179051(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  279nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50455116(CHEMBL2113540)
Affinity DataKi:  292nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]R-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179050(1-(3-chlorophenyl)-3-(9-((2R,3R,4S,5S)-5-(ethylcar...)
Affinity DataKi:  315nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179026(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  319nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179036(1-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydro...)
Affinity DataKi:  324nMAssay Description:Binding affinity against rat adenosine A3 receptor expressed in CHO cells using [125I]-.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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