Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 50036829
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090697(7-Chloro-2-phenyl-[1,8]naphthyridin-4-ol | 7-chlor...)
Affinity DataKi:  0.150nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50118810((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-((R)-1-phenyl...)
Affinity DataKi:  0.600nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090700(7-Bromo-2-phenyl-[1,8]naphthyridin-4-ol | 7-bromo-...)
Affinity DataKi:  0.700nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  1.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50009552(2-[6-Amino-2-(2-morpholin-4-yl-ethylamino)-purin-9...)
Affinity DataKi:  1.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090684(7-Methoxy-2-phenyl-[1,8]naphthyridin-4-ol | 7-meth...)
Affinity DataKi:  1.60nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090709(7-Fluoro-2-phenyl-[1,8]naphthyridin-4-ol | CHEMBL9...)
Affinity DataKi:  4.10nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090691(7-Ethoxy-2-phenyl-[1,8]naphthyridin-4-ol | 7-ethox...)
Affinity DataKi:  5.20nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50059101(2-(4-Fluoro-phenyl)-7-methyl-1H-[1,8]naphthyridin-...)
Affinity DataKi:  5.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090683(7-Amino-2-phenyl-1H-[1,8]naphthyridin-4-one | 7-Am...)
Affinity DataKi:  5.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090705(7-Methyl-2-phenyl-[1,8]naphthyridin-4-ol | 7-methy...)
Affinity DataKi:  5.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  10nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090690(2-(2-Fluoro-phenyl)-7-methyl-[1,8]naphthyridin-4-o...)
Affinity DataKi:  11nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50080398((2R,3S,4R,5R)-2-Hydroxymethyl-5-[6-((S)-1-methyl-2...)
Affinity DataKi:  12nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  14nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  16nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  16nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090708(7-Methyl-2-phenyl-[1,8]naphthyridin-4-ylamine | 7-...)
Affinity DataKi:  17nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50009552(2-[6-Amino-2-(2-morpholin-4-yl-ethylamino)-purin-9...)
Affinity DataKi:  25nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  26nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090701(7-Phenoxy-2-phenyl-[1,8]naphthyridin-4-ol | 7-phen...)
Affinity DataKi:  26nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090704(CHEMBL97624 | Cyclohexyl-(7-methyl-2-phenyl-[1,8]n...)
Affinity DataKi:  28nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  49nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  63nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090700(7-Bromo-2-phenyl-[1,8]naphthyridin-4-ol | 7-bromo-...)
Affinity DataKi:  66nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090685(7-Methyl-2-phenyl-[1,8]naphthyridine-4-thiol | CHE...)
Affinity DataKi:  80nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090697(7-Chloro-2-phenyl-[1,8]naphthyridin-4-ol | 7-chlor...)
Affinity DataKi:  100nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090698((7-Methyl-2-phenyl-[1,8]naphthyridin-4-yl)-hydrazi...)
Affinity DataKi:  100nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090709(7-Fluoro-2-phenyl-[1,8]naphthyridin-4-ol | CHEMBL9...)
Affinity DataKi:  170nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  390nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  418nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090708(7-Methyl-2-phenyl-[1,8]naphthyridin-4-ylamine | 7-...)
Affinity DataKi:  420nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090692(1-Ethyl-7-methyl-2-phenyl-1H-[1,8]naphthyridin-4-o...)
Affinity DataKi:  450nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090705(7-Methyl-2-phenyl-[1,8]naphthyridin-4-ol | 7-methy...)
Affinity DataKi:  460nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  460nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090690(2-(2-Fluoro-phenyl)-7-methyl-[1,8]naphthyridin-4-o...)
Affinity DataKi:  470nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090693(CHEMBL97665 | Dimethyl-(7-methyl-2-phenyl-[1,8]nap...)
Affinity DataKi:  550nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50059101(2-(4-Fluoro-phenyl)-7-methyl-1H-[1,8]naphthyridin-...)
Affinity DataKi:  630nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50009552(2-[6-Amino-2-(2-morpholin-4-yl-ethylamino)-purin-9...)
Affinity DataKi:  750nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090702(7-Methyl-4-phenoxy-2-phenyl-[1,8]naphthyridine | 7...)
Affinity DataKi:  810nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090704(CHEMBL97624 | Cyclohexyl-(7-methyl-2-phenyl-[1,8]n...)
Affinity DataKi:  830nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090689(4-Chloro-7-methyl-2-phenyl-[1,8]naphthyridine | 4-...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CHA from A1 Adenosine receptor of Bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090710(4-(7-Methyl-2-phenyl-[1,8]naphthyridin-4-yl)-piper...)
Affinity DataKi:  1.20E+3nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090685(7-Methyl-2-phenyl-[1,8]naphthyridine-4-thiol | CHE...)
Affinity DataKi:  1.25E+3nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090703(5-Methoxy-1-methyl-7-phenyl-1H-[1,8]naphthyridin-2...)
Affinity DataKi:  1.30E+3nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090684(7-Methoxy-2-phenyl-[1,8]naphthyridin-4-ol | 7-meth...)
Affinity DataKi:  1.40E+3nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090698((7-Methyl-2-phenyl-[1,8]naphthyridin-4-yl)-hydrazi...)
Affinity DataKi:  1.80E+3nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090701(7-Phenoxy-2-phenyl-[1,8]naphthyridin-4-ol | 7-phen...)
Affinity DataKi:  1.90E+3nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50090700(7-Bromo-2-phenyl-[1,8]naphthyridin-4-ol | 7-bromo-...)
Affinity DataKi:  2.10E+3nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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