Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50037646
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175108((5Z,8Z,11Z,14Z)-1-(4-(4-fluorophenyl)piperazin-1-y...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175122(N-(4-methoxyphenyl)oleamide | CHEMBL199960)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175119(N-(3,5-dimethoxyphenethyl)oleamide | CHEMBL199402)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175117(N-(4-methoxybenzyl)oleamide | CHEMBL372530)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175120(N-(4-methoxyphenethyl)oleamide | CHEMBL199702)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175107((5Z,8Z,11Z,14Z)-N-(4-morpholinophenyl)icosa-5,8,11...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175126((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175107((5Z,8Z,11Z,14Z)-N-(4-morpholinophenyl)icosa-5,8,11...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175107((5Z,8Z,11Z,14Z)-N-(4-morpholinophenyl)icosa-5,8,11...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175126((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175126((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175108((5Z,8Z,11Z,14Z)-1-(4-(4-fluorophenyl)piperazin-1-y...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175120(N-(4-methoxyphenethyl)oleamide | CHEMBL199702)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175108((5Z,8Z,11Z,14Z)-1-(4-(4-fluorophenyl)piperazin-1-y...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175120(N-(4-methoxyphenethyl)oleamide | CHEMBL199702)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175114((5Z,8Z,11Z,14Z)-1-(4-(3,4-dimethylphenyl)piperazin...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175134((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxyphenethyl)icosa-5,...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175117(N-(4-methoxybenzyl)oleamide | CHEMBL372530)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175138((5Z,8Z,11Z,14Z)-N-(2,5-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175128((5Z,8Z,11Z,14Z)-N-(4-methoxyphenyl)icosa-5,8,11,14...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175112((5Z,8Z,11Z,14Z)-N-(4-methoxybenzyl)icosa-5,8,11,14...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175117(N-(4-methoxybenzyl)oleamide | CHEMBL372530)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175104((5Z,8Z,11Z,14Z)-1-(4-(4-chlorophenyl)piperazin-1-y...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175119(N-(3,5-dimethoxyphenethyl)oleamide | CHEMBL199402)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175119(N-(3,5-dimethoxyphenethyl)oleamide | CHEMBL199402)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175122(N-(4-methoxyphenyl)oleamide | CHEMBL199960)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175122(N-(4-methoxyphenyl)oleamide | CHEMBL199960)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50054471(cid_6604822 | (5Z,8Z)-Icosa-5,8,11,14-tetraenoic a...)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175105(4-Methoxyphenethylarachidonoylamide | (5Z,8Z,11Z,1...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175121((E)-N-(4-methoxyphenethyl)undec-2-enamide | CHEMBL...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175123((E)-N-(4-methoxyphenyl)undec-2-enamide | CHEMBL198...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175130((E)-N-(3,5-dimethoxyphenethyl)undec-2-enamide | CH...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175137(N-(2,4-dimethoxyphenethyl)docos-13-enamide | CHEMB...)
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175126((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175128((5Z,8Z,11Z,14Z)-N-(4-methoxyphenyl)icosa-5,8,11,14...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175134((5Z,8Z,11Z,14Z)-N-(2,4-dimethoxyphenethyl)icosa-5,...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175138((5Z,8Z,11Z,14Z)-N-(2,5-dimethoxybenzyl)icosa-5,8,1...)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175114((5Z,8Z,11Z,14Z)-1-(4-(3,4-dimethylphenyl)piperazin...)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175107((5Z,8Z,11Z,14Z)-N-(4-morpholinophenyl)icosa-5,8,11...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175112((5Z,8Z,11Z,14Z)-N-(4-methoxybenzyl)icosa-5,8,11,14...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175123((E)-N-(4-methoxyphenyl)undec-2-enamide | CHEMBL198...)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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