Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50040367
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393161BDBM50393161(CHEMBL2153439)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393129BDBM50393129(CHEMBL2153461)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393123BDBM50393123(CHEMBL2153446)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393133BDBM50393133(CHEMBL2153465)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393136BDBM50393136(CHEMBL2153468)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393122BDBM50393122(CHEMBL2153445)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393130BDBM50393130(CHEMBL2153462)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393135BDBM50393135(CHEMBL2153467)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393134BDBM50393134(CHEMBL2153466)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393118BDBM50393118(CHEMBL2153441)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393161BDBM50393161(CHEMBL2153439)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393127BDBM50393127(CHEMBL2153459)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393131BDBM50393131(CHEMBL2153463)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393143BDBM50393143(CHEMBL2153581)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393119BDBM50393119(CHEMBL2153442)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393148BDBM50393148(CHEMBL2153586)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393117BDBM50393117(CHEMBL2153440)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393120BDBM50393120(CHEMBL2153443)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393137BDBM50393137(CHEMBL2153469)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393121BDBM50393121(CHEMBL2153444)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393141BDBM50393141(CHEMBL2153579)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393148BDBM50393148(CHEMBL2153586)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393128BDBM50393128(CHEMBL2153460)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393142BDBM50393142(CHEMBL2153580)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393149BDBM50393149(CHEMBL2153587)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393123BDBM50393123(CHEMBL2153446)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393117BDBM50393117(CHEMBL2153440)
Affinity DataIC50: 115nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393143BDBM50393143(CHEMBL2153581)
Affinity DataIC50: 135nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393158BDBM50393158(CHEMBL2153596)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393156BDBM50393156(CHEMBL2153594)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393157BDBM50393157(CHEMBL2153595)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393150BDBM50393150(CHEMBL2153588)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393138BDBM50393138(CHEMBL2153470)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393140BDBM50393140(CHEMBL2153472)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393147BDBM50393147(CHEMBL2153585)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393126BDBM50393126(CHEMBL2153457)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393145BDBM50393145(CHEMBL2153583)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393132BDBM50393132(CHEMBL2153464)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393158BDBM50393158(CHEMBL2153596)
Affinity DataIC50: 435nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393125BDBM50393125(CHEMBL2153448)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393144BDBM50393144(CHEMBL2153582)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393139BDBM50393139(CHEMBL2153471)
Affinity DataIC50: 720nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393162BDBM50393162(CHEMBL2153436)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393152BDBM50393152(CHEMBL2153590)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393124BDBM50393124(CHEMBL2153447)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393146BDBM50393146(CHEMBL2153584)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393163BDBM50393163(CHEMBL2153438)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target2-oxoglutarate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393123BDBM50393123(CHEMBL2153446)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393159BDBM50393159(CHEMBL2153597)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393162BDBM50393162(CHEMBL2153436)
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in human CHO cells assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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