Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50040971
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403044(CHEMBL179241)
Affinity DataEC50:  3.00E+3nMAssay Description:Increase in CPT1 activity in human MCF7 cells assessed as increase in radiolabeled palmitoylcarnitineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 16nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: 20nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 21nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403041(CHEMBL2216776)
Affinity DataIC50: 26nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403029(CHEMBL2216792)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403042(CHEMBL2216775)
Affinity DataIC50: 65nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: 130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403033(CHEMBL1231507)
Affinity DataIC50: 140nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403041(CHEMBL2216776)
Affinity DataIC50: 150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403043(CHEMBL2216780)
Affinity DataIC50: 190nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403028(CHEMBL2216769)
Affinity DataIC50: 240nMAssay Description:Inhibition of CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403030(CHEMBL2216768)
Affinity DataIC50: 250nMAssay Description:Inhibition of CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403028(CHEMBL2216769)
Affinity DataIC50: 360nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 380nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403029(CHEMBL2216792)
Affinity DataIC50: 700nMAssay Description:Inhibition of rat CPT1A expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 740nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: 800nMAssay Description:Inhibition of CPT2 in 24 hrs fasted rat liver mitochondria assessed as palmitoylcarnitine oxidation by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM80613(SMR000674573 | cid_9926449 | 1-(2,3,4-Trimethoxy-b...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403032(CHEMBL2216785)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403033(CHEMBL1231507)
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitochondrial carnitine/acylcarnitine carrier protein(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403026(CHEMBL2216788)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CACTMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403032(CHEMBL2216785)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403043(CHEMBL2216780)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403046(CHEMBL2216772)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403046(CHEMBL2216772)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50118093((4-Hydroxy-phenyl)-oxo-acetic acid | CHEMBL129918)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of CPT1B in heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403033(CHEMBL1231507)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: 2.73E+4nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403043(CHEMBL2216780)
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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