Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50042363
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313633BDBM50313633(1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)benzyl)ind...)
Affinity DataEC50:  600nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424646BDBM50424646(CHEMBL2313530)
Affinity DataEC50:  1.30E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424645BDBM50424645(CHEMBL2313520)
Affinity DataEC50:  2.40E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424644BDBM50424644(CHEMBL2313515)
Affinity DataEC50:  3.20E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424643BDBM50424643(CHEMBL2313499)
Affinity DataEC50:  3.30E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424641BDBM50424641(CHEMBL2313498)
Affinity DataEC50:  3.30E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424641BDBM50424641(CHEMBL2313498)
Affinity DataEC50:  3.31E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424642BDBM50424642(CHEMBL2313507)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424640BDBM50424640(CHEMBL2313512)
Affinity DataEC50:  5.20E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424639BDBM50424639(CHEMBL2313508)
Affinity DataEC50:  5.60E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424659BDBM50424659(CHEMBL2313519)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424653BDBM50424653(CHEMBL2313495)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424654BDBM50424654(CHEMBL2313531)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424651BDBM50424651(CHEMBL2313497)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424652BDBM50424652(CHEMBL2313496)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424657BDBM50424657(CHEMBL2313506)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424658BDBM50424658(CHEMBL2313504)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424655BDBM50424655(CHEMBL2313529)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424656BDBM50424656(CHEMBL2313510)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424649BDBM50424649(CHEMBL2313514)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424650BDBM50424650(CHEMBL2313513)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424647BDBM50424647(CHEMBL2313517)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424648BDBM50424648(CHEMBL2313516)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed