Compile Data Set for Download or QSAR
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Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50044165
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007206(CHEMBL3237867)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007196(CHEMBL3237864)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007193(CHEMBL3237865)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007207(CHEMBL3237860)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007202(CHEMBL3237868)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  7nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007201(CHEMBL3237870)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007205(CHEMBL3237871)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007209(CHEMBL3237874)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007197(CHEMBL3237869)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007208(CHEMBL3237861)
Affinity DataIC50:  29nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50:  31nMAssay Description:Inhibition of beta5i subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007206(CHEMBL3237867)
Affinity DataIC50:  46nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007204(CHEMBL3237872)
Affinity DataIC50:  54nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50:  59nMAssay Description:Inhibition of beta5i subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50007193(CHEMBL3237865)
Affinity DataIC50:  75nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  76nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  78nMAssay Description:Inhibition of beta5i subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007196(CHEMBL3237864)
Affinity DataIC50:  120nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  120nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007197(CHEMBL3237869)
Affinity DataIC50:  130nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50:  140nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  140nMAssay Description:Inhibition of beta5 subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50:  140nMAssay Description:Inhibition of beta5 subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50:  150nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50:  170nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007201(CHEMBL3237870)
Affinity DataIC50:  210nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007202(CHEMBL3237868)
Affinity DataIC50:  250nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50:  280nMAssay Description:Inhibition of beta5 subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50:  450nMAssay Description:Inhibition of beta5i subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007204(CHEMBL3237872)
Affinity DataIC50:  500nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50432548(LACTACYSTIN)
Affinity DataIC50:  500nMAssay Description:Inhibition of beta5 subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007205(CHEMBL3237871)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of beta5 subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50430990(BELACTOSIN A)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007193(CHEMBL3237865)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007197(CHEMBL3237869)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007196(CHEMBL3237864)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007206(CHEMBL3237867)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50432548(LACTACYSTIN)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of beta5i subunit of immunoproteasome (unknown origin) by active-site ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant cathepsin G (unknown origin) using Suc-Ala-Ala-Pro-Phe-AMC as substrate by spectrofluorometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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