Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50044859
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033089(CHEMBL3342959)
Affinity DataIC50: 0.620nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033094(CHEMBL3342964)
Affinity DataIC50: 0.870nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033083(CHEMBL3342953)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033060(CHEMBL3342952)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033085(CHEMBL3342955)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033085(CHEMBL3342955)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033084(CHEMBL3342954)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033034(CHEMBL3342950)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033091(CHEMBL3342961)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033094(CHEMBL3342964)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033092(CHEMBL3342962)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033092(CHEMBL3342962)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033086(CHEMBL3342956)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033093(CHEMBL3342963)
Affinity DataIC50: 51nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033097(CHEMBL3342945)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033033(CHEMBL3342947)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033093(CHEMBL3342963)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033088(CHEMBL3342958)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033089(CHEMBL3342959)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033087(CHEMBL3342957)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033035(CHEMBL3342951)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033086(CHEMBL3342956)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033087(CHEMBL3342957)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033091(CHEMBL3342961)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033096(CHEMBL285954)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033059(CHEMBL3341770)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033096(CHEMBL285954)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033099(CHEMBL3342949)
Affinity DataIC50: 840nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033084(CHEMBL3342954)
Affinity DataIC50: 890nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033060(CHEMBL3342952)
Affinity DataIC50: 890nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033088(CHEMBL3342958)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033090(CHEMBL3342960)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033083(CHEMBL3342953)
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033097(CHEMBL3342945)
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033090(CHEMBL3342960)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033034(CHEMBL3342950)
Affinity DataIC50: 3.60E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033059(CHEMBL3341770)
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033100(CHEMBL3342948)
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033033(CHEMBL3342947)
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033035(CHEMBL3342951)
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033095(CHEMBL3342946)
Affinity DataIC50: 7.70E+3nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033095(CHEMBL3342946)
Affinity DataIC50: 9.70E+3nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033098(CHEMBL3342944)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in CHO cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed