Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50046812
Affinity DataEC50: 3.40E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 708nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 724nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.37E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.89E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 780nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 888nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.35E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.24E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 332nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.71E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 882nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 559nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.27E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 589nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 603nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 389nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.22E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.75E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.34E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 266nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 363nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu8 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Positive allosteric modulation of mGlu5 in rat astrocytesMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu6 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu4 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu3 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu2 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu1 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Positive allosteric modulation of rat mGlu5 assessed as calcium mobilization by cell-based assayMore data for this Ligand-Target Pair
