Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50046812
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132604(CHEMBL3633979)
Affinity DataEC50:  3.40E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132613(CHEMBL3633969)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132612(CHEMBL3633970)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132543(CHEMBL3633971)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132545(CHEMBL3633972)
Affinity DataEC50:  708nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132611(CHEMBL3633973)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132610(CHEMBL3633974)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132546(CHEMBL3633975)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132548(CHEMBL3633976)
Affinity DataEC50:  724nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132609(CHEMBL3633977)
Affinity DataEC50:  794nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132607(CHEMBL3633978)
Affinity DataEC50:  5.37E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132665(CHEMBL3633968)
Affinity DataEC50:  3.89E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132601(CHEMBL3634189)
Affinity DataEC50:  780nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132598(CHEMBL3634190)
Affinity DataEC50:  888nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132591(CHEMBL3634191)
Affinity DataEC50:  1.35E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132590(CHEMBL3634192)
Affinity DataEC50:  3.24E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50:  360nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132520(CHEMBL3633944)
Affinity DataEC50:  332nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132519(CHEMBL3633945)
Affinity DataEC50:  1.71E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132518(CHEMBL3633946)
Affinity DataEC50:  882nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132512(CHEMBL3633947)
Affinity DataEC50:  559nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132670(CHEMBL3633958)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132669(CHEMBL3633964)
Affinity DataEC50:  1.27E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132668(CHEMBL3633965)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132665(CHEMBL3633968)
Affinity DataEC50:  3.90E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132589(CHEMBL3633952)
Affinity DataEC50:  1.12E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132588(CHEMBL3633953)
Affinity DataEC50:  589nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132587(CHEMBL3633954)
Affinity DataEC50:  603nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132586(CHEMBL3633955)
Affinity DataEC50:  389nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132562(CHEMBL3633956)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132559(CHEMBL3633957)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132511(CHEMBL3633948)
Affinity DataEC50:  1.22E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132557(CHEMBL3633959)
Affinity DataEC50:  2.75E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132555(CHEMBL3633960)
Affinity DataEC50:  257nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132553(CHEMBL3633961)
Affinity DataEC50:  2.34E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132552(CHEMBL3633962)
Affinity DataEC50:  266nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132549(CHEMBL3633963)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132669(CHEMBL3633964)
Affinity DataEC50:  1.26E+3nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132668(CHEMBL3633965)
Affinity DataEC50: <1.00E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132667(CHEMBL3633966)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132666(CHEMBL3633967)
Affinity DataEC50: <3.16E+4nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50:  363nMAssay Description:Positive allosteric modulation of human mGlu5 expressed in HEK293 cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 8(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu8 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50:  360nMAssay Description:Positive allosteric modulation of mGlu5 in rat astrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 6(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu6 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu4 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 3(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu3 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu2 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of mGlu1 receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50132507(CHEMBL3633943)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of rat mGlu5 assessed as calcium mobilization by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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