Compile Data Set for Download or QSAR
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Report error Found 3 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 1893
TargetMitogen-activated protein kinase 14(Human)
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14831(3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-(4-chl...)
Affinity DataKd:  1.16E+3nMpH: 7.0 T: 23°CAssay Description:The exchange curve assays were run as two half-reactions using an SLM Aminco Bowman Series 2 model SQ-340 fluorescence detector. In the first half re...More data for this Ligand-Target Pair
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MMDB
PDB3D3D Structure (crystal)

TargetMitogen-activated protein kinase 14(Human)
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  0.100nMpH: 7.0 T: 23°CAssay Description:The exchange curve assays were run as two half-reactions using an SLM Aminco Bowman Series 2 model SQ-340 fluorescence detector. In the first half re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetMitogen-activated protein kinase 14(Human)
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14832(3-(4-fluorophenyl)-2-pyridin-4-yl-6-thia-1,4-diaza...)
Affinity DataKd:  180nMpH: 7.0 T: 23°CAssay Description:The exchange curve assays were run as two half-reactions using an SLM Aminco Bowman Series 2 model SQ-340 fluorescence detector. In the first half re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed