BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50000957

Bromodomain-containing protein 1(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL

BDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)

IC50: 1.68E+3nMAssay Description:Inhibition of human BRD4 BD1 (67 to 152 residues) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Purchase CHEMBL MCE
PC cid PC sid PDB Similars

Details Article PubMed PDB

3D Structure (crystal)