Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50005095
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50: 20nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488029((S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 190nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488030((R,S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 210nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488028((R)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 950nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143314(CHEMBL298826 | (+)-Epibatidine | 2-(6-Chloro-pyrid...)
Affinity DataIC50: 1.34E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143320(2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]hept...)
Affinity DataIC50: 2.79E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50: 1.19E+4nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82068(Nicotine-D salicylate | CHEMBL9732 | Nicotine-L sa...)
Affinity DataIC50: 4.22E+5nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed