Compile Data Set for Download or QSAR
Found 27 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50008260
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517212(CHEMBL4463449)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517209(CHEMBL4561516)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517208(CHEMBL4577891)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517194(CHEMBL4460559)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517196(CHEMBL4564535)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517193(CHEMBL4438749)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517211(CHEMBL4450797)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517206(CHEMBL4469210)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517201(CHEMBL4539507)
Affinity DataIC50:  4.20E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50062727(CHEMBL3397721)
Affinity DataIC50:  4.30E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517203(CHEMBL4467078)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517213(CHEMBL4557705)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517207(CHEMBL4440578)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517197(CHEMBL4579845)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517205(CHEMBL4448302)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517202(CHEMBL4516607)
Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517195(CHEMBL4460064)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517216(CHEMBL4546295)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517199(CHEMBL4436200)
Affinity DataIC50:  8.40E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517198(CHEMBL4558793)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517217(CHEMBL4550568)
Affinity DataIC50:  9.50E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517192(CHEMBL4533671)
Affinity DataIC50:  9.60E+3nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517214(CHEMBL4532632)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517215(CHEMBL4440852)
Affinity DataIC50:  1.31E+4nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517204(CHEMBL4528757)
Affinity DataIC50:  1.51E+4nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517210(CHEMBL4438177)
Affinity DataIC50:  1.58E+4nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fraunhofer Institute for Molecular Biology and Applied Ecology IME

Curated by ChEMBL
LigandPNGBDBM50517200(CHEMBL4465395)
Affinity DataIC50:  2.39E+4nMAssay Description:Antagonist actvity in pFA-GAL4-DBD fused PPARgamma LBD (unknown origin) transfected in HEK293T cells assessed as inhibition of rosiglitazone-induced ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed