Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50017885
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109368BDBM50109368(CHEMBL3601212)
Affinity DataIC50: 14nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006932BDBM50006932(CHEMBL3237245)
Affinity DataIC50: 29nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 561983BDBM561983(US11396496, Compound A1 | BDBM50369389)
Affinity DataIC50: 60nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50120422BDBM50120422(CHEMBL3617852)
Affinity DataIC50: 61nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130557BDBM50130557(CHEMBL3632882)
Affinity DataIC50: 85nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200467BDBM50200467(CHEMBL3899754)
Affinity DataIC50: 140nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593788BDBM50593788(CHEMBL5172581)
Affinity DataIC50: 575nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605859BDBM50605859(CHEMBL5207192)
Affinity DataIC50: 677nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605861BDBM50605861(CHEMBL5195422)
Affinity DataIC50: 805nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605858BDBM50605858(CHEMBL5203566)
Affinity DataIC50: 815nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006931BDBM50006931(CHEMBL2402207)
Affinity DataIC50: 940nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605862BDBM50605862(CHEMBL5189014)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605860BDBM50605860(CHEMBL5174036)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593790BDBM50593790(CHEMBL5173969)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109403BDBM50109403(CHEMBL3600394)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50076479BDBM50076479(CHEMBL3235901)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
University College London

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605864BDBM50605864(CHEMBL5181288)
Affinity DataIC50: 2.93E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed