Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50020243
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211650(3-(4-(4-((1-(2-chlorocyclopent-1-enyl)ethoxy)carbo...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211648(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211655(4-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211647(3-(4-(4-((1-(2-chlorocyclohex-1-enyl)ethoxy)carbon...)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211646(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211649(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211651(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211653(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211654(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211645(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)-3-met...)
Affinity DataIC50:  510nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211652(3-{2'-[1-(2-chloro-phenyl)-ethoxycarbonylamino]-bi...)
Affinity DataIC50: >4.00E+4nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed