Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50021832
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228359(CHEMBL254815 | methyl 2-chloro-6,8-dihydroxy-9-{1-...)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228361(2-chloro-6,8-dihydroxy-1-methoxy-3,9-dimethyltetra...)
Affinity DataIC50:  4.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228358(CHEMBL253120 | methyl 2-chloro-9-ethyl-6,8-dihydro...)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed