Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50033992
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50344100(2-((2R)-1-((4-methylphenyl)sulfonyl)-3-oxo-2-piper...)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355063(CHEMBL1834619)
Affinity DataKi:  0.300nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355062(CHEMBL1834752)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355057(CHEMBL1834751)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355064(CHEMBL1834616)
Affinity DataKi:  0.900nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355056(CHEMBL1834614)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355058(CHEMBL1834750)
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355059(CHEMBL1834620)
Affinity DataKi:  3.10nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355060(CHEMBL1834615)
Affinity DataKi:  3.5nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50244617((2R,3S)-2,3-dihydroxy-N-((R)-6-(piperidin-1-ylmeth...)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355061(CHEMBL1834618)
Affinity DataKi:  4.70nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355065(CHEMBL1835761)
Affinity DataKi:  18nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355066(CHEMBL1835767)
Affinity DataKi:  29nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355067(CHEMBL1835763)
Affinity DataKi:  35nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355068(CHEMBL1835766)
Affinity DataKi:  52nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355069(CHEMBL1835756)
Affinity DataKi:  64nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355070(CHEMBL1834749)
Affinity DataKi:  69.9nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355071(CHEMBL1835769)
Affinity DataKi:  98nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355072(CHEMBL1835760)
Affinity DataKi:  159nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355073(CHEMBL1835757)
Affinity DataKi:  183nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355074(CHEMBL1834617)
Affinity DataKi:  198nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355075(CHEMBL1835768)
Affinity DataKi:  214nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355076(CHEMBL1835753)
Affinity DataKi:  296nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355077(CHEMBL1835755)
Affinity DataKi:  311nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355078(CHEMBL1835758)
Affinity DataKi:  331nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355079(CHEMBL1834613)
Affinity DataKi:  418nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355080(CHEMBL1835754)
Affinity DataKi:  565nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355081(CHEMBL1835765)
Affinity DataKi:  614nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355082(CHEMBL1835752)
Affinity DataKi:  1.68E+3nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataKi:  6.37E+3nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355084(CHEMBL1835759)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50355085(CHEMBL1835764)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed