Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50036406
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369097BDBM50369097(CHEMBL604851)
Affinity DataEC50:  164nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453346BDBM50453346(CHEMBL2113449)
Affinity DataEC50:  167nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369104BDBM50369104(CHEMBL604026)
Affinity DataEC50:  306nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369091BDBM50369091(CHEMBL604019)
Affinity DataEC50:  322nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369084BDBM50369084(CHEMBL604440)
Affinity DataEC50:  358nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369112BDBM50369112(CHEMBL603812)
Affinity DataEC50:  415nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369113BDBM50369113(CHEMBL606318)
Affinity DataEC50:  840nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369103BDBM50369103(CHEMBL603809)
Affinity DataEC50:  877nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369100BDBM50369100(CHEMBL606319)
Affinity DataEC50:  3.14E+3nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454091BDBM50454091(CHEMBL2113450)
Affinity DataEC50:  6.48E+3nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369102BDBM50369102(CHEMBL605265)
Affinity DataEC50:  7.16E+3nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085658BDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataEC50:  8.20E+3nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369110BDBM50369110(CHEMBL605685)
Affinity DataEC50:  8.53E+3nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369108BDBM50369108(CHEMBL605691)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369105BDBM50369105(CHEMBL606315)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369094BDBM50369094(CHEMBL604023)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369093BDBM50369093(CHEMBL603389)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369096BDBM50369096(CHEMBL605264)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369087BDBM50369087(CHEMBL605065)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369109BDBM50369109(CHEMBL605056)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369099BDBM50369099(CHEMBL605690)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369095BDBM50369095(CHEMBL605057)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369092BDBM50369092(CHEMBL604234)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369098BDBM50369098(CHEMBL605055)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369111BDBM50369111(CHEMBL604849)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 35804BDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369088BDBM50369088(CHEMBL604649)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453224BDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369107BDBM50369107(CHEMBL603596)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369085BDBM50369085(CHEMBL603602)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369106BDBM50369106(CHEMBL603808)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50205705BDBM50205705((2S,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369090BDBM50369090(CHEMBL605478)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369089BDBM50369089(CHEMBL605473)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  5.48E+4nMAssay Description:Functional activity against adenosine A1 receptor from rat atria.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed