Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50040734
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399165(CHEMBL2180137)
Affinity DataIC50: 189nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399163(CHEMBL2180139)
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50: 1.38E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399175(CHEMBL2180171)
Affinity DataIC50: 1.78E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 1.87E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399164(CHEMBL2180138)
Affinity DataIC50: 2.28E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399166(CHEMBL2180136)
Affinity DataIC50: 2.35E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399190(CHEMBL2180149)
Affinity DataIC50: 2.44E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399200(CHEMBL2180148)
Affinity DataIC50: 2.49E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399161(CHEMBL2180141)
Affinity DataIC50: 2.64E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399172(CHEMBL2180174)
Affinity DataIC50: 2.69E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399197(CHEMBL2180151)
Affinity DataIC50: 3.39E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399160(CHEMBL2180142)
Affinity DataIC50: 3.93E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399188(CHEMBL2180183)
Affinity DataIC50: 4.11E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399187(CHEMBL2180184)
Affinity DataIC50: 4.29E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399186(CHEMBL2180185)
Affinity DataIC50: 5.29E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399203(CHEMBL451082)
Affinity DataIC50: 5.97E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399177(CHEMBL2180169)
Affinity DataIC50: 9.54E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399196(CHEMBL2180152)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399195(CHEMBL2180153)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399194(CHEMBL2180154)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399193(CHEMBL2180155)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399198(CHEMBL229357)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399192(CHEMBL2180156)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399191(CHEMBL2180157)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399199(CHEMBL2180150)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399159(CHEMBL2180144)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399206(CHEMBL2180180)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399184(CHEMBL2180159)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399182(CHEMBL2180164)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399181(CHEMBL2180165)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399180(CHEMBL2180166)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399162(CHEMBL2180140)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399178(CHEMBL2180168)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399176(CHEMBL2180170)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399168(CHEMBL2180178)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399189(CHEMBL2180182)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399170(CHEMBL2180176)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399202(CHEMBL484675)
Affinity DataIC50: 1.03E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399169(CHEMBL2180177)
Affinity DataIC50: 1.07E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399185(CHEMBL2180158)
Affinity DataIC50: 1.08E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399201(CHEMBL2180147)
Affinity DataIC50: 1.18E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399171(CHEMBL2180175)
Affinity DataIC50: 1.24E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50370141(TNP-ATP)
Affinity DataIC50: 1.52E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399173(CHEMBL2180173)
Affinity DataIC50: 1.74E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399205(CHEMBL2180181)
Affinity DataIC50: 2.32E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399174(CHEMBL2180172)
Affinity DataIC50: 2.46E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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