Compile Data Set for Download or QSAR
Found 236 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 9268
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454208((Z)-3-fluoro-4-(3-(4-fluorophenyl)-1H- indol-1-yl)...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454208((Z)-3-fluoro-4-(3-(4-fluorophenyl)-1H- indol-1-yl)...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454209((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454209((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454210((Z)-4-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454210((Z)-4-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454211((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454211((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454212((Z)-methyl 1-(4-amino-2-fluorobut-2-en- 1-yl)-3-(3...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454212((Z)-methyl 1-(4-amino-2-fluorobut-2-en- 1-yl)-3-(3...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454213((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454213((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454214((Z)-methyl 1-(4-amino-2-fluorobut-2-en- 1-yl)-3-(3...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454214((Z)-methyl 1-(4-amino-2-fluorobut-2-en- 1-yl)-3-(3...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454215((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454215((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454216((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454216((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454217((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454217((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454218((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454218((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454219((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454219((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454220((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454220((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454221((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-2- methyl-3-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454221((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-2- methyl-3-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454222((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454222((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454223((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(dimet...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454223((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(dimet...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454224((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-2-met...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454224((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-2-met...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454225((Z)-1-(4-amino-2-fluorobut-2-en-l-yl)-2- methyl-3-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454225((Z)-1-(4-amino-2-fluorobut-2-en-l-yl)-2- methyl-3-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454226((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(5-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454226((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(5-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454227((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (5-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454227((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (5-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454228((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454228((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (3-(N,N-d...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454229((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454229((Z)-ethyl 1-(4-amino-2-fluorobut-2-en-1- yl)-3-(3-...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454230((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (4-fluoro...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454230((Z)-1-(4-amino-2-fluorobut-2-en-1-yl)-3- (4-fluoro...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454231(US10717733, Compound 24 | US11098045, Compound 24 ...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454231(US10717733, Compound 24 | US11098045, Compound 24 ...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOxidized low-density lipoprotein receptor 1(Bovine)
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454232((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: >300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis Ltd.

US Patent
LigandPNGBDBM454232((Z)-3-(1-(4-amino-2-fluorobut-2-en-1-yl)- 2-methyl...)
Affinity DataIC50: <300nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
In DepthDetails US Patent
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