Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 9388
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals, Inc.

US Patent
LigandPNGBDBM463328( [3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-(2-pyrrol...)
Affinity DataIC50:  1.10nMAssay Description:Radioligand binding assays for human 5-HT2A receptor was conducted using the 5-HT2 agonist [125I]DOI as radioligand. To define nonspecific binding, 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals, Inc.

US Patent
LigandPNGBDBM463330(1-(3-Acetyl-phenyl)-3-[3-(2-methyl-2H-pyrazol-3-yl...)
Affinity DataIC50:  5nMAssay Description:Radioligand binding assays for human 5-HT2A receptor was conducted using the 5-HT2 agonist [125I]DOI as radioligand. To define nonspecific binding, 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals, Inc.

US Patent
LigandPNGBDBM463329(1-(4-Chloro-benzyl)-3-[3-(2-methyl-2H-pyrazol-3-yl...)
Affinity DataIC50:  10.2nMAssay Description:Radioligand binding assays for human 5-HT2A receptor was conducted using the 5-HT2 agonist [125I]DOI as radioligand. To define nonspecific binding, 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals, Inc.

US Patent
LigandPNGBDBM463331(2-(4-Fluoro-phenyl)-N-[3-(2-methyl-2H-pyrazol-3-yl...)
Affinity DataIC50:  13.7nMAssay Description:Radioligand binding assays for human 5-HT2A receptor was conducted using the 5-HT2 agonist [125I]DOI as radioligand. To define nonspecific binding, 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent