Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for assayid = 11 entry = 50025054
Target5-hydroxytryptamine receptor 2C(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031942BDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10755BDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  20nMAssay Description:Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234920BDBM50234920(Barettin | cyclo[(6-bromo-8-entryptophan)arginine]...)
Affinity DataKi:  340nMAssay Description:Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241836BDBM50241836(cyclo[(6-bromotryptophan)arginine] | CHEMBL511609)
Affinity DataKi:  4.63E+3nMAssay Description:Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed