Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50001212
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272471BDBM50272471(CHEMBL4127540)
Affinity DataIC50: 110nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272473BDBM50272473(CHEMBL4126588)
Affinity DataIC50: 171nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272481BDBM50272481(CHEMBL4128940)
Affinity DataKi:  274nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272482BDBM50272482(CHEMBL4130151)
Affinity DataIC50: 350nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272487BDBM50272487(CHEMBL4126157)
Affinity DataIC50: 356nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272484BDBM50272484(CHEMBL4129458)
Affinity DataKi:  814nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272471BDBM50272471(CHEMBL4127540)
Affinity DataKi:  876nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272483BDBM50272483(CHEMBL4128794)
Affinity DataIC50: 1.87E+3nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50272482BDBM50272482(CHEMBL4130151)
Affinity DataKi:  4.68E+3nMAssay Description:Displacement of [3H]8-prazosin from adrenergic alpha1 receptor in Wistar rat cortex incubated for 30 mins by microbeta liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed