Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50002842
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM43362(TETRAMETHYLTHIURAM DISULFIDE | SMR000059023 | MLS0...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463618(CHEMBL4241062)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463622(CHEMBL4245637)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463615(CHEMBL4251179)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463620(CHEMBL4240937)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50366038(CHEMBL1356238)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463621(CHEMBL3144916)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463617(CHEMBL4238380)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463616(CHEMBL4241417)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463619(CHEMBL4242081)
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463614(CHEMBL4237334)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50463613(CHEMBL1927732)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProtein-lysine 6-oxidase(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed