Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50003791
LigandChemical structure of BindingDB Monomer ID 50476002BDBM50476002(CHEMBL217511)
Affinity DataEC50:  0.676nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475982BDBM50475982(CHEMBL215375)
Affinity DataEC50:  19nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50062397BDBM50062397(N''-cyano-N-(1,1-dimethylpropyl)-N'-pyridin-3-ylgu...)
Affinity DataEC50:  22nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475961BDBM50475961(CHEMBL214841)
Affinity DataEC50:  29nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50044253BDBM50044253(CHEMBL11684 | (3S,4R)-3-hydroxy-2,2-dimethyl-4-(2-...)
Affinity DataEC50:  35nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475954BDBM50475954(CHEMBL216256)
Affinity DataEC50:  55nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475963BDBM50475963(CHEMBL2062142 | WAY-133537)
Affinity DataEC50:  102nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475985BDBM50475985(CHEMBL424909)
Affinity DataEC50:  129nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50476001BDBM50476001(CHEMBL387063)
Affinity DataEC50:  245nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 86249BDBM86249(ZD-6169 | ZD 6169)
Affinity DataEC50:  295nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50475975BDBM50475975(CHEMBL386843)
Affinity DataEC50:  331nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed