Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50007308
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000727BDBM50000727((R)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-di...)
Affinity DataEC50:  0.0780nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061108BDBM50061108(3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimeth...)
Affinity DataEC50:  0.208nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061113BDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataEC50:  0.790nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061111BDBM50061111((R)-3-(1,1-Dimethyl-heptyl)-6,6,9-trimethyl-6a,7,8...)
Affinity DataEC50:  1nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061116BDBM50061116(3-(1,1-Dimethyl-heptyl)-1-hydroxy-9-methyl-benzo[c...)
Affinity DataEC50:  4.60nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061114BDBM50061114(3-(1,1-Dimethyl-heptyl)-1-hydroxy-6,6-dimethyl-6H-...)
Affinity DataEC50:  5.40nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061110BDBM50061110(1-Acetoxy-3-(1,1-dimethyl-heptyl)-6,6-dimethyl-6H-...)
Affinity DataEC50:  39nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061118BDBM50061118(3-(1,1-Dimethyl-heptyl)-1-hydroxy-6,6-dimethyl-6a,...)
Affinity DataEC50:  116nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Science

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061117BDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  261nMAssay Description:Effective concentration for inhibition of human Cannabinoid receptor 2-mediated adenylyl cyclase using African green monkey (COS-7) cells transfected...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed