Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50007518
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510090(CHEMBL4535730)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510091(CHEMBL4519542)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510092(CHEMBL4593987)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510094(CHEMBL4460072)
Affinity DataEC50:  991nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair