Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50017704
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185450BDBM50185450(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(5,6...)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185470BDBM50185470(3-(benzo[d][1,3]dioxol-5-yl)-4-(5-(2-(5,6,7,8-tetr...)
Affinity DataIC50: 1.03nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185464BDBM50185464(3-(benzo[d][1,3]dioxol-5-yl)-4-(3-(2-(5,6,7,8-tetr...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185469BDBM50185469(3-(benzo[d][1,3]dioxol-5-yl)-4-(3-(2-(1-methyl-1,2...)
Affinity DataIC50: 1.47nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185457BDBM50185457(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-benzyl-5-(2-(5,6...)
Affinity DataIC50: 1.84nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185456BDBM50185456(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(5,6...)
Affinity DataIC50: 1.86nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185452BDBM50185452(3-(benzo[d][1,3]dioxol-5-yl)-4-(5-(2-(5,6,7,8-tetr...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185468BDBM50185468(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(1-m...)
Affinity DataIC50: 2.58nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185467BDBM50185467(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-butyl-5-(2-(5,6,...)
Affinity DataIC50: 3nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185463BDBM50185463(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-phenyl-5-(2-(5,6...)
Affinity DataIC50: 3.27nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185462BDBM50185462(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(5,6...)
Affinity DataIC50: 5.43nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185459BDBM50185459(3-(benzo[d][1,3]dioxol-5-yl)-4-(3-(3-(4,5-dihydro-...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185458BDBM50185458(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(6-(...)
Affinity DataIC50: 11nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185451BDBM50185451(3-(benzo[d][1,3]dioxol-5-yl)-4-(3-(2-(6-(methylami...)
Affinity DataIC50: 17.5nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185453BDBM50185453(3-(2-(4-chlorophenyl)thiazol-5-yl)-4-(1-methyl-5-(...)
Affinity DataIC50: 18nMAssay Description:Inhibition of alpha-v-beta-5 integrin in 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed