Compile Data Set for Download or QSAR
Found 51 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50017774
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186291(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186278(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186270(2-benzyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tet...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186290(3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186269(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186309(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186292(2-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186306(3-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186316(2-(phenylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186283(2-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186293(7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydrois...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186311(3-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186296(2-(cyclohexylmethyl)-6-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  1.01nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186281((6-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquino...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186295(2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186285(CHEMBL208829 | N-isopropyl-7-(3-(piperidin-1-yl)pr...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186286(1-(phenylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186305(2-(phenylsulfonyl)-6-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186273((7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquino...)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186300(1-(7-(3-(piperidin-1-yl)propoxy)-1,2,4,5-tetrahydr...)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186275(3-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2...)
Affinity DataKi:  12.1nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186284(2-(cyclohexylmethyl)-5-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  15.4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186297(CHEMBL209099 | N-isopropyl-7-(3-(piperidin-1-yl)pr...)
Affinity DataKi:  17.1nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186289(1-(phenylsulfonyl)-6-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186277(1-(7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoqui...)
Affinity DataKi:  19.4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186279((7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroquinolin...)
Affinity DataKi:  22.6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186288(2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  23.8nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186268(1-(cyclohexylmethyl)-6-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186312(1-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186287(CHEMBL377975 | N-isopropyl-7-(3-(piperidin-1-yl)pr...)
Affinity DataKi:  42.3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186272(6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroqu...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186307(2-(cyclohexylmethyl)-8-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186276(2-ethyl-5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  84.2nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186308(2-ethyl-8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  95.2nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186314(7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroqu...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186313(1-(cyclohexylmethyl)-5-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186315(8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydrois...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186299(1-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186318(1-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186304(5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroqu...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186303(8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroqu...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186302((8-(3-(piperidin-1-yl)propoxy)-3,4-dihydroquinolin...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186301(1-(phenylsulfonyl)-8-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186298(2-(phenylsulfonyl)-5-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186310((5-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquino...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186282(2-(phenylsulfonyl)-8-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186280((8-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquino...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186274(5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydrois...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186317(1-ethyl-8-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186271(1-ethyl-5-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi: >300nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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