Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50040850
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50241132(7-(3-Hydroxy-2-phenyl-propionyloxy)-9,9-dimethyl-3...)
Affinity DataKi:  0.170nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50326219(CHEMBL1242950 | CHEMBL2206334 | 4-(4-butylpiperidi...)
Affinity DataKi:  891nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50401038(CHEMBL2206335)
Affinity DataKi:  1.29E+3nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50149891(CHEMBL360055 | 2,2',2''-[1,2,3-BENZENE-TRIYLTRIS(O...)
Affinity DataKi:  8.51E+3nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50401037(BRUCINE)
Affinity DataKi:  4.47E+4nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed