Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50035248
TargetAcetylcholinesterase(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataEC50:  43nMAssay Description:In vitro reversal of vecuronium-induced neuromuscular block in guinea pig hemi-diaphragm.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50117577(1-Benzyl-4-[3-(5,6-dimethoxy-benzo[b]thiophen-2-yl...)
Affinity DataEC50:  19nMAssay Description:In vitro reversal of vecuronium-induced neuromuscular block in guinea pig hemi-diaphragm.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50117574(1-Benzyl-1-methyl-4-[3-(5-methyl-1-phenyl-1H-pyraz...)
Affinity DataEC50:  430nMAssay Description:In vitro reversal of vecuronium-induced neuromuscular block in guinea pig hemi-diaphragm.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50117576(1-Benzyl-4-[3-(6-methoxy-naphthalen-2-yl)-3-oxo-pr...)
Affinity DataEC50:  530nMAssay Description:In vitro reversal of vecuronium-induced neuromuscular block in guinea pig hemi-diaphragm.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed