Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50049017
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232938BDBM50232938(CHEMBL4088509)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21281BDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232936BDBM50232936(CHEMBL4071738)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232941BDBM50232941(CHEMBL4084087)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232940BDBM50232940(CHEMBL4071007)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232933BDBM50232933(CHEMBL4094388)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232937BDBM50232937(CHEMBL4086649)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399157BDBM50399157(CHEMBL2179724)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232934BDBM50232934(CHEMBL4098746)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232935BDBM50232935(CHEMBL4102128)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232942BDBM50232942(CHEMBL4077875)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232939BDBM50232939(CHEMBL4104545)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232944BDBM50232944(CHEMBL4094331)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Sassari

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232943BDBM50232943(CHEMBL4090242)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed