Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50000502
TargetMuscarinic acetylcholine receptor M1(Rat)
Novo Nordisk Cns Division

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003363BDBM50003363(1-Methyl-5-(4-pentylsulfanyl-[1,2,5]thiadiazol-3-y...)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity against M1 receptor from rat hippocampus, using [3H]oxotremorine-M (Oxo-M) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Novo Nordisk Cns Division

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003363BDBM50003363(1-Methyl-5-(4-pentylsulfanyl-[1,2,5]thiadiazol-3-y...)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity against M1 receptor from rat hippocampus, using [3H]oxotremorine-M (Oxo-M) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed