Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50043727
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50445222(CHEMBL3105228)
Affinity DataIC50: 790nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M5 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50445224(CHEMBL3105213)
Affinity DataIC50: 1.10E+3nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M5 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50445223(CHEMBL3105208)
Affinity DataIC50: 2.10E+3nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M5 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50445225(CHEMBL1459098)
Affinity DataIC50: 5.67E+3nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M5 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed