Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50046079
TargetCytochrome P450 2C8(Homo sapiens (Human))
Eisai Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50029064(CHEMBL3343259)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using rosiglitazone as susbtrate incubated for 30 mins prior to substrate addition for 10 mins by LC-M...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Eisai Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50093793(E-2006 | Lemborexant)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using rosiglitazone as susbtrate incubated for 30 mins prior to substrate addition for 10 mins by LC-M...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed