Compile Data Set for Download or QSAR
Found 22 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50046160
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.150nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097043(CHEMBL3580910)
Affinity DataKi:  0.450nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096976(CHEMBL3580908)
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096973(CHEMBL3580907)
Affinity DataKi:  3.80nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096968(CHEMBL3580919)
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096977(CHEMBL3580909)
Affinity DataKi:  4.90nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM30707(2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097066(CHEMBL3580915)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096971(CHEMBL3580926)
Affinity DataKi:  17nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097064(CHEMBL3580913)
Affinity DataKi:  44nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097067(CHEMBL3580917)
Affinity DataKi:  68nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097068(CHEMBL3580918)
Affinity DataKi:  160nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataKi:  190nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096969(CHEMBL3580924)
Affinity DataKi:  220nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097050(CHEMBL3580912)
Affinity DataKi:  498nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097116(CHEMBL3580921)
Affinity DataKi:  530nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097115(CHEMBL3580920)
Affinity DataKi:  535nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097117(CHEMBL3580922)
Affinity DataKi:  560nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097118(CHEMBL3580923)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50096970(CHEMBL3580925)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097048(CHEMBL3580911)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50097065(CHEMBL3580914)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed