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Found 8 Enz. Inhib. hit(s) with all data for assayid = 7 entry = 50017915
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50188381(5-iodo-1-(naphthalen-2-ylmethyl)indoline-2,3-dione...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50055220(1-Benzyl-2,3-dioxo-2,3-dihydro-1H-indole-5-carboxy...)
Affinity DataKi:  1.26E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50188383(1-butyl-2,3-dioxoindoline-5-carboxamide | CHEMBL37...)
Affinity DataKi:  1.91E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50133617(1-Benzyl-5-iodo-1H-indole-2,3-dione | 1-benzyl-5-i...)
Affinity DataKi:  5.01E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50188384(1-butyl-5-iodoindoline-2,3-dione | CHEMBL209287 | ...)
Affinity DataKi:  6.61E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50055216(1-Methyl-2,3-dioxo-2,3-dihydro-1H-indole-5-carboxy...)
Affinity DataKi:  7.24E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50055218(1-(2-naphthlmethyl) isatin-5-carboxamide | 1-Napht...)
Affinity DataIC50:  370nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1a(Human SARS coronavirus (SARS-CoV))
Peking University

Curated by ChEMBL
LigandPNGBDBM50188382(2,3-dioxo-1-propylindoline-5-carboxamide | CHEMBL2...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of SARS CoV 3C-like proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed