Affinity DataKi: 60nM ΔG°: -41.2kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataKi: 170nM ΔG°: -38.6kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataKi: 320nM ΔG°: -37.1kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nM ΔG°: -32.7kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nM ΔG°: -30.8kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nM ΔG°: -27.1kJ/molepH: 7.5 T: 2°CAssay Description:HSP90 inhibitors identified using Fluorescence resonance energy transfer assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMpH: 7.4Assay Description:To assess the affinity of compounds binding to Hsp90, we measured their ability to compete with the binding of a fluorescent analog of GA (GM-Bodipy)...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair
Affinity DataIC50: <20nMpH: 7.4Assay Description:The fluorescent labeled small molecule used in the present invention was VER-00051001 (synthesized by reference to the synthetic method described in ...More data for this Ligand-Target Pair