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Found 38 of ph data with Target = 'MAP kinase-interacting serine/threonine-protein kinase 1'
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181594(US9139577, 4.100 | US9708274, 4.100)
Affinity DataIC50:  14nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181612(US9139577, 4.118 | US9708274, 4.118)
Affinity DataIC50:  21nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181400(US9139577, 2.008 | US9708274, 2.008)
Affinity DataIC50:  25nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181632(US9139577, 4.138 | US9708274, 4.138)
Affinity DataIC50:  27nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM261870(US9708274, 4.136)
Affinity DataIC50:  29nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181410(US9139577, 2.018 | US9708274, 2.018)
Affinity DataIC50:  34nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181380(US9139577, 1.011 | US9708274, 1.011)
Affinity DataIC50:  34nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98040(US8486953, 53)
Affinity DataIC50:  35nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181582(US9139577, 4.088 | US9708274, 4.088)
Affinity DataIC50:  36nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181568(US9139577, 4.074 | US9708274, 4.074)
Affinity DataIC50:  38nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181649(US9139577, 5.008 | US9708274, 5.008)
Affinity DataIC50:  39nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181439(US9139577, 2.048 | US9708274, 2.048)
Affinity DataIC50:  40nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM261908(US9708274, 7.010)
Affinity DataIC50:  40nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181401(US9139577, 2.009 | US9708274, 2.009)
Affinity DataIC50:  49nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM261907(US9708274, 7.009)
Affinity DataIC50:  50nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181528(US9139577, 4.034 | US9708274, 4.034)
Affinity DataIC50:  51nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181493(US9139577, 3.054 | US9708274, 3.054)
Affinity DataIC50:  51nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181385(US9139577, 1.016 | US9708274, 1.016)
Affinity DataIC50:  53nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181388(US9139577, 1.019 | US9708274, 1.019)
Affinity DataIC50:  54nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181565(US9139577, 4.071 | US9708274, 4.071)
Affinity DataIC50:  55nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181440(US9139577, 3.001 | US9708274, 3.001)
Affinity DataIC50:  60nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181645(US9139577, 5.004 | US9708274, 5.004)
Affinity DataIC50:  66nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181488(US9139577, 3.049 | US9708274, 3.049)
Affinity DataIC50:  68nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181398(US9139577, 2.006 | US9708274, 2.006)
Affinity DataIC50:  71nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181470(US9139577, 3.031 | US9708274, 3.031)
Affinity DataIC50:  75nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181552(US9139577, 4.058 | US9708274, 4.058)
Affinity DataIC50:  75nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181478(US9139577, 3.039 | US9708274, 3.039)
Affinity DataIC50:  77nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98034(US8486953, 9)
Affinity DataIC50:  100nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98032(US8486953, 2)
Affinity DataIC50:  120nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181662(US9139577, 7.006 | US9708274, 7.006)
Affinity DataIC50:  164nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98033(US8486953, 6)
Affinity DataIC50:  180nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98035(US8486953, 10)
Affinity DataIC50:  210nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98038(US8486953, 41)
Affinity DataIC50:  210nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM181393(US9139577, 2.001 | US9708274, 2.001)
Affinity DataIC50:  228nMpH: 7.5Assay Description:The inhibition of kinase activity of MNK1a was assessed using pre-activated GST-MNK1a. The 2xMKNK1 (MNK1) mixture is prepared in 50 mM HEPES pH 7.5, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98041(US8486953, 71)
Affinity DataIC50:  400nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98039(US8486953, 48)
Affinity DataIC50:  460nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98036(US8486953, 19)
Affinity DataIC50:  590nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec International

US Patent
LigandPNGBDBM98037(US8486953, 34)
Affinity DataIC50:  680nMpH: 7.4Assay Description:In vitro kinase assay using human Mnk1 and Mnk2.More data for this Ligand-Target Pair
In DepthDetails US Patent