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Found 23 of ph data with Target = 'Nuclear receptor subfamily 5 group A member 2'
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22373((3aS,6aR)-5-[(4E)-oct-4-en-4-yl]-N,4-diphenyl-1,2,...)
Affinity DataEC50:  430nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22395(N-[(3aS,6aR)-5-hexyl-4-phenyl-1,2,3,3a,6,6a-hexahy...)
Affinity DataEC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22375((3aS,6aR)-4-butyl-5-[(4E)-oct-4-en-4-yl]-N-phenyl-...)
Affinity DataEC50:  22nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22376((3aS,6aR)-4-cyclohexyl-5-[(4E)-oct-4-en-4-yl]-N-ph...)
Affinity DataEC50:  12nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
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TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22377((3aS,6aR)-4-(4-bromophenyl)-5-[(4E)-oct-4-en-4-yl]...)
Affinity DataEC50:  160nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22378((3aS,6aR)-4-(3-methoxyphenyl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  100nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22379((3aS,6aR)-4-(naphthalen-2-yl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  60nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22380((3aS,6aR)-5-[(3E)-hex-3-en-3-yl]-N,4-diphenyl-1,2,...)
Affinity DataEC50:  1.40E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22381((3aS,6aR)-5-[(6E)-dodec-6-en-6-yl]-N,4-diphenyl-1,...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22382((3aS,6aR)-5-(hexan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  70nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22383((3aS,6aR)-5-(decan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  320nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22384((3aS,6aR)-5-methyl-N,4-diphenyl-1,2,3,3a,6,6a-hexa...)
Affinity DataEC50:  2.10E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22385((3aS,6aR)-5-hexyl-N,4-diphenyl-1,2,3,3a,6,6a-hexah...)
Affinity DataEC50:  34nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22386((3aS,6aR)-5-cyclohexyl-N,4-diphenyl-1,2,3,3a,6,6a-...)
Affinity DataEC50:  230nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22387((3aS,6aR)-5-dodecyl-N,4-diphenyl-1,2,3,3a,6,6a-hex...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22388((3aS,6aR)-N,4,5-triphenyl-1,2,3,3a,6,6a-hexahydrop...)
Affinity DataEC50:  150nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22389((3aS,6aR)-N-(3-fluorophenyl)-5-hexyl-4-phenyl-1,2,...)
Affinity DataEC50:  330nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22390((3aS,6aR)-N-(4-chlorophenyl)-5-hexyl-4-phenyl-1,2,...)
Affinity DataEC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22391((3aS,6aR)-N-(2,3-dimethylphenyl)-5-hexyl-4-phenyl-...)
Affinity DataEC50:  30nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22392((3aS,6aR)-5-hexyl-4-phenyl-N-[4-(trifluoromethoxy)...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22393((3aS,6aR)-N-(4-tert-butylphenyl)-5-hexyl-4-phenyl-...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22394((3aS,6aR)-5-hexyl-N-(4-iodophenyl)-4-phenyl-1,2,3,...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22374((3aS,6aR)-4-methyl-5-[(4E)-oct-4-en-4-yl]-N-phenyl...)
Affinity DataEC50:  90nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed