Compile Data Set for Download or QSAR
maximum 50k data
Found 20 of ph data with Target = 'Orotate phosphoribosyltransferase'
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214779(OPRT inhibitor, 2)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214785(OPRT inhibitor, 8)
Affinity DataKi:  170nM ΔG°:  -38.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214778(OPRT inhibitor, 1 )
Affinity DataKi:  190nM ΔG°:  -38.4kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214791(OPRT inhibitor, 14)
Affinity DataKi:  220nM ΔG°:  -38.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214786(OPRT inhibitor, 9)
Affinity DataKi:  270nM ΔG°:  -37.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214784(OPRT inhibitor, 7)
Affinity DataKi:  270nM ΔG°:  -37.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214782(OPRT inhibitor, 5)
Affinity DataKi:  300nM ΔG°:  -37.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214780(OPRT inhibitor, 3)
Affinity DataKi:  350nM ΔG°:  -36.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214783(OPRT inhibitor, 6)
Affinity DataKi:  350nM ΔG°:  -36.8kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214781(OPRT inhibitor, 4)
Affinity DataKi:  370nM ΔG°:  -36.7kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214790(OPRT inhibitor, 13)
Affinity DataKi:  470nM ΔG°:  -36.1kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214793(OPRT inhibitor, 16)
Affinity DataKi:  480nM ΔG°:  -36.1kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214796(OPRT inhibitor, 19)
Affinity DataKi:  500nM ΔG°:  -36.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214792(OPRT inhibitor, 15)
Affinity DataKi:  500nM ΔG°:  -36.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214797(OPRT inhibitor, 20)
Affinity DataKi:  510nM ΔG°:  -35.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214795(OPRT inhibitor, 18)
Affinity DataKi:  570nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214787(OPRT inhibitor, 10)
Affinity DataKi:  690nM ΔG°:  -35.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214794(OPRT inhibitor, 17)
Affinity DataKi:  750nM ΔG°:  -35.0kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214788(OPRT inhibitor, 11)
Affinity DataKi:  1.30E+3nM ΔG°:  -33.6kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrotate phosphoribosyltransferase(Plasmodium falciparum)
Albert Einstein College Of Medicine

LigandPNGBDBM214789(OPRT inhibitor, 12)
Affinity DataKi:  1.55E+4nM ΔG°:  -27.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition constants (Ki, equivalent to Kd for competitive inhibitors) were measured at 25 °C by adding purified OPRT enzymes (25 nM for PfOPRT a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed