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Found 1733 of ph data with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform'
LigandPNGBDBM50403098(CHEMBL2216893 | US8754089, 4-amino-6-(((1S)-1-(6-m...)
Affinity DataKi:  5nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124086(US8754089, 4-amino-6-(((1S)-1-(4-oxo-3-phenyl-4H-p...)
Affinity DataKi:  8.20nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124095(US8754089, 4-amino-6-((1-(6-methyl-4-oxo-3-(2-pyri...)
Affinity DataKi:  10.8nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124096(US8754089, 4-amino-6-((1-(6-methyl-4-oxo-3-phenyl-...)
Affinity DataKi:  12.6nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124083(US8754089, 4-amino-6-(((1S)-1-(3-(3-fluorophenyl)-...)
Affinity DataKi:  15.7nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124094(US8754089, 4-amino-6-((1-(4-oxo-3-phenyl-4H-pyrido...)
Affinity DataKi:  15.9nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124087(US8754089, 4-amino-6-(((1S)-1-(6-methyl-4-oxo-3-(2...)
Affinity DataKi:  21.4nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124077(US10428087, Example 72 | US10829502, Example 72 | ...)
Affinity DataKi:  23.1nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124079(US10428087, Example 70 | US10829502, Example 70 | ...)
Affinity DataKi:  27.7nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124090(US8754089, 4-amino-6-((1-(3-(3,5-difluorophenyl)-6...)
Affinity DataKi:  33nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM124085(US8754089, 4-amino-6-(((1S)-1-(4-oxo-3-(2-pyridiny...)
Affinity DataKi:  42.4nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124088(US8754089, 4-amino-6-((1-(3-(2-(methylsulfonyl)phe...)
Affinity DataKi:  52.8nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124091(US8754089, 4-amino-6-((1-(3-(3-fluorophenyl)-4-oxo...)
Affinity DataKi:  57.1nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124082(US8754089, 4-amino-6-(((1S)-1-(3-(3,5-difluorophen...)
Affinity DataKi:  63.7nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124097(US8754089, 6-methyl-2-(1-(9H-purin-6-ylamino)ethyl...)
Affinity DataKi:  80.2nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124074(US8754089, 2-((4-amino-3-iodo-1H-pyrazolo[3,4-d]py...)
Affinity DataKi:  84.9nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM124089(US8754089, 4-amino-6-((1-(3-(3,5-difluorophenyl)-4...)
Affinity DataKi:  89nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124093(US8754089, 4-amino-6-((1-(4-oxo-3-(2-pyridinyl)-4H...)
Affinity DataKi:  104nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124103(US8754089, 7-fluoro-3-(3-fluorophenyl)-2-((1S)-1-(...)
Affinity DataKi:  110nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124100(US8754089, 7-fluoro-2-((1S)-1-(9H-purin-6-ylamino)...)
Affinity DataKi:  184nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124084(US8754089, 4-amino-6-(((1S)-1-(3-(4-methyl-2-pyrid...)
Affinity DataKi:  230nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124104(US8754089, 7-fluoro-3-(3-fluorophenyl)-2-(1-(9H-pu...)
Affinity DataKi:  360nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124092(US8754089, 4-amino-6-((1-(3-(4-methyl-2-pyridinyl)...)
Affinity DataKi:  471nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM124101(US8754089, 7-fluoro-2-(1-(9H-purin-6-ylamino)ethyl...)
Affinity DataKi:  659nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124078(US8754089, 3-(3-fluorophenyl)-6-methyl-2-((9H-puri...)
Affinity DataKi:  711nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124076(US10428087, Example 71 | US10829502, Example 71 | ...)
Affinity DataKi:  802nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124075(US8754089, 2-((6-amino-9H-purin-9-yl)methyl)-6-met...)
Affinity DataKi:  6.28E+3nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM124081(US8754089, 4-amino-6-(((1R)-1-(4-oxo-3-phenyl-4H-p...)
Affinity DataKi:  6.32E+3nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124098(US8754089, 6-methyl-3-(2-methylphenyl)-2-((9H-puri...)
Affinity DataKi:  9.71E+3nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM124102(US8754089, 7-fluoro-3-(3-fluorophenyl)-2-((1R)-1-(...)
Affinity DataKi:  1.98E+4nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124099(US8754089, 7-fluoro-2-((1R)-1-(9H-purin-6-ylamino)...)
Affinity DataKi:  2.15E+4nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM124080(US8754089, 4-amino-6-(((1R)-1-(3-(2-(methylsulfony...)
Affinity DataKi:  2.46E+4nMpH: 7.0Assay Description:A PI3K Alphascreen assay (PerkinElmer, Waltham, Mass.) was used to measure the activity of a panel of four phosphoinositide 3-kinases: PI3Kα, PI...More data for this Ligand-Target Pair
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LigandPNGBDBM172655(US9090628, 315 | US9090628, 316)
Affinity DataIC50: <0.0350nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172706(US9090628, 366)
Affinity DataIC50: <0.0350nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172707(US9090628, 367)
Affinity DataIC50:  0.0480nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM172459(US9090628, 101 | US9090628, 102 | US9090628, 103 |...)
Affinity DataIC50:  0.102nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172459(US9090628, 101 | US9090628, 102 | US9090628, 103 |...)
Affinity DataIC50:  0.106nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172459(US9090628, 101 | US9090628, 102 | US9090628, 103 |...)
Affinity DataIC50:  0.107nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172682(US9090628, 342)
Affinity DataIC50:  0.160nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172654(US9090628, 314 | US9090628, 318 | US9090628, 320)
Affinity DataIC50:  0.178nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172654(US9090628, 314 | US9090628, 318 | US9090628, 320)
Affinity DataIC50:  0.236nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172588(US9090628, 248 | US9090628, 309 | US9090628, 310)
Affinity DataIC50:  0.262nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172686(US9090628, 346 | US9090628, 348)
Affinity DataIC50:  0.288nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172606(US9090628, 266 | US9090628, 287 | US9090628, 288)
Affinity DataIC50:  0.292nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172619(US9090628, 279 | US9090628, 291 | US9090628, 292)
Affinity DataIC50:  0.293nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172700(US9090628, 360 | US9090628, 361)
Affinity DataIC50:  0.311nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172665(US9090628, 325)
Affinity DataIC50:  0.313nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172693(US9090628, 353 | US9090628, 355)
Affinity DataIC50:  0.314nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172619(US9090628, 279 | US9090628, 291 | US9090628, 292)
Affinity DataIC50:  0.324nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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LigandPNGBDBM172654(US9090628, 314 | US9090628, 318 | US9090628, 320)
Affinity DataIC50:  0.335nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
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