Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ph data with Target = 'Plasmepsin I'
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

LigandPNGBDBM8025((2S)-N-[(2S,3S)-4-{[(1S)-2-(4-bromophenyl)-1-carba...)
Affinity DataKi:  98nM ΔG°:  -39.6kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme activities were assayed by monitoring the hydrolysis of substrate in the presence or absence of inhibitor compounds. The hydrolysis was record...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

LigandPNGBDBM8022((2S)-N-[(2S,3S)-4-{[(S)-carbamoyl(phenyl)methyl]am...)
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme activities were assayed by monitoring the hydrolysis of substrate in the presence or absence of inhibitor compounds. The hydrolysis was record...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

LigandPNGBDBM8023((2S)-N-[(2S,3S)-4-{[(1S)-1-carbamoyl-2-phenylethyl...)
Affinity DataKi:  2.10E+3nM ΔG°:  -32.1kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme activities were assayed by monitoring the hydrolysis of substrate in the presence or absence of inhibitor compounds. The hydrolysis was record...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

LigandPNGBDBM8021((2S)-2-{[(2S,3S)-2-hydroxy-3-[(2S)-3-methyl-2-(pyr...)
Affinity DataKi:  2.90E+3nM ΔG°:  -31.3kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme activities were assayed by monitoring the hydrolysis of substrate in the presence or absence of inhibitor compounds. The hydrolysis was record...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

LigandPNGBDBM8024((2R,5S,6R)-3-Aza-2-benzyl-5-hydroxy-7-phenyl-6-[(p...)
Affinity DataKi:  8.00E+3nM ΔG°:  -28.8kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme activities were assayed by monitoring the hydrolysis of substrate in the presence or absence of inhibitor compounds. The hydrolysis was record...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed